Heider F.; Pantsar T.; Kudolo M.; Ansideri F.; De Simone A.; Pruccoli L.; Schneider T.; Goettert M.I.; Tarozzi A.; Andrisano V.; Laufer S.A.; Koch P., Pyridinylimidazoles as GSK3β Inhibitors: The Impact of Tautomerism on Compound Activity via Water Networks, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 1407 - 1414 [articolo]
Morroni Fabiana, Sita Giulia, Djemil Alice, D'Amico Massimo, Pruccoli Letizia, Cantelli-Forti Giorgio, Hrelia Patrizia, Tarozzi Andrea., Comparison of Adaptive Neuroprotective Mechanisms of Sulforaphane and its Interconversion Product Erucin in in Vitro and in Vivo Models of Parkinson's Disease, «JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY», 2018, 66, pp. 856 - 865 [articolo]Open Access
Dias Viegas, Flávia Pereira; de Freitas Silva, Matheus; Divino da Rocha, Miguel; Castelli, Maísa Rosa; Riquiel, Mariana Máximo; Machado, Rafael Pereira; Vaz, Sarah Macedo; Simões de Lima, Laís Medeiros; Mancini, Karla Cristine; Marques de Oliveira, Patrícia Cruz; Morais, Élida Parreira; Gontijo, Vanessa Silva; da Silva, Fernanda Motta R.; D'Alincourt da Fonseca Peçanha, Dora; Castro, Newton Gonçalves; Neves, Gilda A.; Giusti-Paiva, Alexandre; Vilela, Fabiana Cardoso; Orlandi, Lidiane; Camps, Ihosvany; Veloso, Márcia Paranho; Leomil Coelho, Luis Felipe; Ionta, Marisa; Ferreira-Silva, Guilherme Álvaro; Pereira, Rodrigo Machado; Dardenne, Laurent E.; Guedes, Isabella Alvim; de Oliveira Carneiro Junior, Wellerson; Quaglio Bellozi, Paula Maria; Pinheiro de Oliveira, Antônio Carlos; Ferreira, Fábio Furlan; Pruccoli, Letizia; Tarozzi, Andrea; Viegas, Claudio*, Design, synthesis and pharmacological evaluation of N-benzyl-piperidinyl-aryl-acylhydrazone derivatives as donepezil hybrids: Discovery of novel multi-target anti-alzheimer prototype drug candidates, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2018, 147, pp. 48 - 65 [articolo]Open Access
Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, Ignacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease, «MOLECULES», 2018, 23, Article number: 1902, pp. 1 - 22 [articolo]Open Access
de Freitas Silva M, Pruccoli L, Morroni F, Sita G, Seghetti F, Viegas C, Tarozzi A, The Keap1/Nrf2-ARE pathway as a pharmacological target for chalcones, «MOLECULES», 2018, 23, Article number: 1803, pp. 1 - 22 [articolo]Open Access
Rampa, Angela; Montanari, Serena; Pruccoli, Letizia; Bartolini, Manuela; Falchi, Federico; Feoli, Alessandra; Cavalli, Andrea; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Chalcone-based carbamates for Alzheimer's disease treatment, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 749 - 764 [articolo]
Dias, Kris Simone T.; de Paula, Cynthia T.; dos Santos, Thiago; Souza, Isis N.O.; Boni, Marina S.; Guimarães, Marcos J.R.; da Silva, Fernanda M.R.; Castro, Newton G.; Neves, Gilda A.; Veloso, Clarice C.; Coelho, Márcio M.; de Melo, Ivo Souza F.; Giusti, Fabiana C.V.; Giusti-Paiva, Alexandre; da Silva, Marcelo L.; Dardenne, Laurent E.; Guedes, Isabella A.; Pruccoli, Letizia; Morroni, Fabiana; Tarozzi, Andrea; Viegas, Claudio*, Design, synthesis and evaluation of novel feruloyl-donepezil hybrids as potential multitarget drugs for the treatment of Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 130, pp. 440 - 457 [articolo]Open Access
Maestri, Valentina; Tarozzi, Andrea; Simoni, Elena; Cilia, Antonio; Poggesi, Elena; Naldi, Marina; Nicolini, Benedetta; Pruccoli, Letizia; Rosini, Michela; Minarini, Anna, Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 136, pp. 259 - 269 [articolo]
Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A., Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 117, pp. 283 - 291 [articolo]
Montanari, Serena; Bartolini, Manuela; Neviani, Paolo; Belluti, Federica; Gobbi, Silvia; Pruccoli, Letizia; Tarozzi, Andrea; Falchi, Federico; Andrisano, Vincenza; Miszta, Przemysław; Cavalli, Andrea; Filipek, Sławomir; Bisi, Alessandra; Rampa, Angela, Multitarget Strategy to Address Alzheimer's Disease: Design, Synthesis, Biological Evaluation, and Computational Studies of Coumarin-Based Derivatives, «CHEMMEDCHEM», 2016, 11, pp. 1296 - 1308 [articolo]Open Access
Rampa, Angela; Tarozzi, Andrea; Mancini, Francesca; Pruccoli, Letizia; Di Martino, Rita Maria Concetta; Gobbi, Silvia; Bisi, Alessandra; De Simone, Angela; Palomba, Francesco; Zaccheroni, Nelsi; Belluti, Federica, Naturally inspired molecules as multifunctional agents for Alzheimer's disease treatment, «MOLECULES», 2016, 21, Article number: 643, pp. 1 - 16 [articolo]Open Access