Foto del docente

Elisa Uliassi

Senior assistant professor (fixed-term)

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Publications

Exertier, Cécile; Salerno, Alessandra; Antonelli, Lorenzo; Fiorillo, Annarita; Ocello, Riccardo; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Masetti, Matteo; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Ilari, Andrea; Bolognesi, Maria Laura, Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis, «JOURNAL OF MEDICINAL CHEMISTRY», 2024, 67, pp. 402 - 419 [Scientific article]Open Access

Pasieka, Anna; Diamanti, Eleonora; Uliassi, Elisa; Laura Bolognesi, Maria, Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?, «CHEMMEDCHEM», 2023, 18, Article number: e202300422 , pp. 1 - 17 [Scientific article]Open Access

Guardigni M.; Pruccoli L.; Santini A.; Simone A.D.; Bersani M.; Spyrakis F.; Frabetti F.; Uliassi E.; Andrisano V.; Pagliarani B.; Fernández-Gómez P.; Palomo V.; Bolognesi M.L.; Tarozzi A.; Milelli A., PROTAC-Induced Glycogen Synthase Kinase 3β Degradation as a Potential Therapeutic Strategy for Alzheimer’s Disease, «ACS CHEMICAL NEUROSCIENCE», 2023, 14, pp. 1963 - 1970 [Scientific article]Open Access

Uliassi, E; Bergamini, C; Rizzardi, N; Naldi, M; Cores, A; Bartolini, M; Menéndez, JC; Bolognesi, ML, Quinolinetrione-tacrine hybrids as multi-target-directed ligands against Alzheimer's disease, «BIOORGANIC & MEDICINAL CHEMISTRY», 2023, 91, Article number: 117419 , pp. 1 - 9 [Scientific article]Open Access

Rocío Marisol Espinoza Chávez; Salerno A.; Liuzzi A.; Ilari A.; Milelli A.; Uliassi E.; Bolognesi M.L., Targeted Protein Degradation for Infectious Diseases: from Basic Biology to Drug Discovery, «ACS BIO & MED CHEM AU», 2023, 3, pp. 32 - 45 [Scientific article]Open Access

Salerno, Alessandra; Seghetti, Francesca; Caciolla, Jessica; Uliassi, Elisa; Testi, Eleonora; Guardigni, Melissa; Roberti, Marinella; Milelli, Andrea; Bolognesi, Maria Laura, Enriching Proteolysis Targeting Chimeras with a Second Modality: When Two Are Better Than One, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 9507 - 9530 [Scientific article]Open Access

Lauriola A.; Uliassi E.; Santucci M.; Bolognesi M.L.; Mor M.; Scalvini L.; Elisi G.M.; Gozzi G.; Tagliazucchi L.; Marverti G.; Ferrari S.; Losi L.; D'Arca D.; Costi M.P., Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing Library, «PHARMACEUTICS», 2022, 14, Article number: 391 , pp. 1 - 22 [Scientific article]Open Access

Albertini, C; Salerno, A; Atzenti, S; Uliassi, E; Massenzio, F; Maruca, A; Rocca, R; Mecava, M; Silva, FSG; Mena, D; Valente, P; Duarte, AI; Chavarria, D; Bissaro, M; Moro, S; Federico, S; Spalluto, G; Soukup, O; Borges, F; Alcaro, S; Monti, B; Oliveira, PJ; Menendez, JC; Bolognesi, ML, Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis, «ACS CHEMICAL NEUROSCIENCE», 2022, 13, pp. 2252 - 2260 [Scientific article]Open Access

Bianco M.D.C.A.D.; Inacio Leite D.; Silva Castelo Branco F.; Boechat N.; Uliassi E.; Bolognesi M.L.; Bastos M.M., The Use of Zidovudine Pharmacophore in Multi-Target-Directed Ligands for AIDS Therapy, «MOLECULES», 2022, 27, Article number: 8502 , pp. 8502 - 8523 [Scientific article]Open Access

Uliassi, Elisa; Nikolic, Lea; Bolognesi, Maria Laura; Legname, Giuseppe, Therapeutic strategies for identifying small molecules against prion diseases, «CELL & TISSUE RESEARCH», 2022, x, pp. 1 - 11 [Scientific article]

Uliassi E.; de Oliveira A.S.; Nascente L.C.; Romeiro L.A.S.; Bolognesi M.L., Cashew nut shell liquid (Cnsl) as a source of drugs for alzheimer’s disease, «MOLECULES», 2021, 26, Article number: 5441 , pp. 1 - 21 [Scientific article]Open Access

Ramos, GD; de Oliveira, AS; Bartolini, M; Naldi, M; Liparulo, I; Bergamini, C; Uliassi, E; Wu, L; Fraser, PE; Abreu, M; Kiametis, AS; Gargano, R; Silveira, ER; Brand, GD; Prchal, L; Soukup, O; Korabecny, J; Bolognesi, ML; Romeiro, LAS, Discovery of sustainable drugs for Alzheimer's disease: cardanol-derived cholinesterase inhibitors with antioxidant and anti-amyloid properties, «RSC MEDICINAL CHEMISTRY», 2021, 12, pp. 1154 - 1163 [Scientific article]Open Access

Gorecki L.; Uliassi E.; Bartolini M.; Janockova J.; Hrabinova M.; Hepnarova V.; Prchal L.; Muckova L.; Pejchal J.; Karasova J.Z.; Mezeiova E.; Benkova M.; Kobrlova T.; Soukup O.; Petralla S.; Monti B.; Korabecny J.; Bolognesi M.L., Phenothiazine-Tacrine Heterodimers: Pursuing Multitarget Directed Approach in Alzheimer's Disease, «ACS CHEMICAL NEUROSCIENCE», 2021, 12, pp. 1698 - 1715 [Scientific article]

Espro C.; Paone E.; Mauriello F.; Gotti R.; Uliassi E.; Bolognesi M.L.; Rodriguez-Padron D.; Luque R., Sustainable production of pharmaceutical, nutraceutical and bioactive compounds from biomass and waste, «CHEMICAL SOCIETY REVIEWS», 2021, 50, pp. 11191 - 11207 [Scientific article]

Perone R.; Albertini C.; Uliassi E.; Di Pietri F.; de Sena Murteira Pinheiro P.; Petralla S.; Rizzardi N.; Fato R.; Pulkrabkova L.; Soukup O.; Tramarin A.; Bartolini M.; Bolognesi M.L., Turning Donepezil into a Multi-Target-Directed Ligand through a Merging Strategy, «CHEMMEDCHEM», 2021, 16, pp. 187 - 198 [Scientific article]Open Access

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