Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R., Design, synthesis and biological activity of some 4-DAMP- related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1995, 5, pp. 2325 - 2330 [articolo]
Chiarini A.; Budriesi R.; Bolognesi M.L.; Minarini A.; Melchiorre C., In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors, «BRITISH JOURNAL OF PHARMACOLOGY», 1995, 114, pp. 1507 - 1517 [articolo]
Melchiorre C.; Minarini A.; Budriesi R.; Chiarini A.; Spampinato S.; Tumiatti V., The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists, «LIFE SCIENCES», 1995, 56, pp. 837 - 844 [articolo]
Minarini A.; Bolognesi M.L.; Budriesi R.; Canossa M.; Chiarini A.; Spampinato S.; Melchiorre C., Design, Synthesis, and Biological Activity of Methoctramine-Related Tetraamines Bearing an 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Moiety: Structural Requirements for Optimum Occupancy of Muscarinic Receptor Subtypes As Revealed by Symmetrical and Unsymmetrical Polyamines, «JOURNAL OF MEDICINAL CHEMISTRY», 1994, 37, pp. 3363 - 3372 [articolo]
Melchiorre C.; Bolognesi M.L.; Chiarini A.; Minarini A.; Spampinato S., Synthesis and Biological Activity of Some Methoctramine-Related Tetraamines Bearing a 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]-benzodiazepin-6-one Moiety as Antimuscarinics: A Second Generation of Highly Selective M2 Muscarinic Receptor Antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1993, 36, pp. 3734 - 3737 [articolo]
Tumiatti V.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R.; Bolognesi M.L., Affinity and selectivity at M2 and M3 muscarinic receptor subtypes of cyclic and open oxygenated analogues of 4-DAMP, «IL FARMACO», 1992, 47, pp. 1133 - 1147 [articolo]
Minarini A.; Budriesi R.; Chiarini A.; Melchiorre C.; Tumiatti V., Further investigation on methoctramine-related tetraamines: Effects of terminal N-substitution and of chain length separating the four nitrogens on M2 muscarinic receptor blocking activity, «IL FARMACO», 1991, 46, pp. 1167 - 1178 [articolo]
Chiarini A.; Minarini A.; Budriesi R.; Melchiorre C., Molecular properties of the histamine H2-receptor. Covalent inhibition by tetraamine disulfides, «IL FARMACO», 1990, 45, pp. 1001 - 1011 [articolo]