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Anna Minarini

Professoressa ordinaria

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Direttrice Scuola di Specializzazione in Farmacia Ospedaliera (nuovo ordinamento)

Pubblicazioni

Melchiorre C.; Angeli P.; Bolognesi M.L.; Chiarini A.; Giardina D.; Gulini U.; Leonardi A.; Marucci G.; Minarini A.; Pigini M.; Quaglia W.; Rosini M.; Tumiatti V., α1-Adrenoreceptor antagonists bearing a quinazoline or a benzodioxane moiety, «PHARMACEUTICA ACTA HELVETIAE», 2000, 74, pp. 181 - 190 [articolo]

Rosini M.; Budriesi R.; Bixel M.G.; Bolognesi M.L.; Chiarini A.; Hucho F.; Krogsgaard-Larsen P.; Mellor I.R.; Minarini A.; Tumiatti V.; Usherwood P.N.R.; Melchiorre C., Design, synthesis, and biological evaluation of symmetrically and unsymmetrically substituted methoctramine-related polyamines as muscular nicotinic receptor noncompetitive antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 5212 - 5223 [articolo]

Bolognesi M.L.; Budriesi R.; Cavalli A.; Chiarini A.; Gotti R.; Leonardi A.; Minarini A.; Poggesi E.; Recanatini M.; Rosini M.; Tumiatti V.; Melchiorre C., WB 4101-related compounds. 2. Role of the ethylene chain separating amine and phenoxy units on the affinity for α1-adrenoreceptor subtypes and 5-HT(1A) receptors, «JOURNAL OF MEDICINAL CHEMISTRY», 1999, 42, pp. 4214 - 4224 [articolo]

Barbier P.; Colelli A.; Bolognesi M.L.; Minarini A.; Tumiatti V.; Corsini G.U.; Melchiorre C.; Maggio R., Antagonist binding profile of the split chimeric muscarinic m2-trunc/m3-tail receptor, «EUROPEAN JOURNAL OF PHARMACOLOGY», 1998, 355, pp. 267 - 274 [articolo]

Melchiorre C.; Bolognesi M.L.; Budriesi R.; Chiarini A.; Giardina D.; Minarini A.; Quaglia W.; Leonardi A., Search for selective antagonists at α1-adrenoreceptors: Neutral or negative antagonism?, «IL FARMACO», 1998, 53, pp. 278 - 286 [articolo]

Minarini A.; Budriesi R.; Chiarini A.; Leonardi A.; Melchiorre C., Search for α1-adrenoceptor subtypes selective antagonists: Design, synthesis and biological activity of cystazosin, an α(1D)-adrenoceptor antagonist, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1998, 8, pp. 1353 - 1358 [articolo]

Bolognesi M.L.; Minarini A.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Spampinato S.; Tumiatti V.; Melchiorre C., Universal template approach to drug design: Polyamines as selective muscarinic receptor antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1998, 41, pp. 4150 - 4160 [articolo]

Melchiorre C.; Angeli P.; Bolognesi M.L.; Budriesi R.; Cacciaguerra S.; Chiarini A.; Crucianelli M.; Giardina D.; Gulini U.; Marucci G.; Minarini A.; Spampinato S.; Tumiatti V., Tetraamines as lead compounds for the design of neurotransmitter receptor ligands:Focus on α-adrenergic and muscarinic receptors recognition, «perspective in receptor research», 1996, 24, pp. 321 - 336 [articolo]

Melchiorre C.; Minarini A.; Spampinato S.; Tumiatti V., Design, synthesis and biological activity of some tetraamines related to methoctramine and 4-DAMP, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1995, 5, pp. 785 - 790 [articolo]

Tumiatti V.; Santi S.; Recanatini M.; Minarini A.; Melchiorre C.; Chiarini A.; Budriesi R., Design, synthesis and biological activity of some 4-DAMP- related compounds, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 1995, 5, pp. 2325 - 2330 [articolo]

Chiarini A.; Budriesi R.; Bolognesi M.L.; Minarini A.; Melchiorre C., In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors, «BRITISH JOURNAL OF PHARMACOLOGY», 1995, 114, pp. 1507 - 1517 [articolo]

Melchiorre C.; Minarini A.; Budriesi R.; Chiarini A.; Spampinato S.; Tumiatti V., The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists, «LIFE SCIENCES», 1995, 56, pp. 837 - 844 [articolo]

Maggio R.; Barbier P.; Bolognesi M.L.; Minarini A.; Tedeschi D.; Melchiorre C., Binding profile of the selective muscarinic receptor antagonist tripitramine, «EUROPEAN JOURNAL OF PHARMACOLOGY-MOLECULAR PHARMACOLOGY SECTION», 1994, 268, pp. 459 - 462 [articolo]

Minarini A.; Bolognesi M.L.; Budriesi R.; Canossa M.; Chiarini A.; Spampinato S.; Melchiorre C., Design, Synthesis, and Biological Activity of Methoctramine-Related Tetraamines Bearing an 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Moiety: Structural Requirements for Optimum Occupancy of Muscarinic Receptor Subtypes As Revealed by Symmetrical and Unsymmetrical Polyamines, «JOURNAL OF MEDICINAL CHEMISTRY», 1994, 37, pp. 3363 - 3372 [articolo]

Melchiorre C.; Bolognesi M.L.; Chiarini A.; Minarini A.; Spampinato S., Synthesis and Biological Activity of Some Methoctramine-Related Tetraamines Bearing a 11-Acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]-benzodiazepin-6-one Moiety as Antimuscarinics: A Second Generation of Highly Selective M2 Muscarinic Receptor Antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 1993, 36, pp. 3734 - 3737 [articolo]