Foto del docente

Andrea Tarozzi

Full Professor

Department for Life Quality Studies

Academic discipline: BIO/14 Pharmacology

Publications

Cindy Juliet Cristancho Ortiz; Caio Miranda Damasio; Letizia Pruccoli; Nathália Fonseca Nadur; Luciana Luiza de Azevedo; Isabella Alvim Guedes; Laurent Emmanuel Dardenne; Arthur Eugen Kümmerle; Andrea Tarozzi; Claudio Viegas Jr, Cinnamoyl-N-Acylhydrazone-Donepezil Hybrids: Synthesis and Evaluation of Novel Multifunctional Ligands Against Neurodegenerative Diseases, «NEUROCHEMICAL RESEARCH», 2020, 45, pp. 3003 - 3020 [Scientific article]

Matheus de Freitas Silva; Ellen Tardelli Lima; Letizia Pruccoli; Newton G Castro; Marcos Jorge R Guimarães; Fernanda M R da Silva; Nathalia Fonseca Nadur; Luciana Luiz de Azevedo; Arthur Eugen Kümmerle; Isabella Alvim Guedes; Laurent Emmanuel Dardenne; Vanessa Silva Gontijo; Andrea Tarozzi; Claudio Viegas, Design, Synthesis and Biological Evaluation of Novel Triazole N-acylhydrazone Hybrids for Alzheimer's Disease, «MOLECULES», 2020, 25, Article number: 3165 , pp. 1 - 18 [Scientific article]Open Access

Andreev S.; Pantsar T.; El-gokha A.; Ansideri F.; Kudolo M.; Anton D.B.; Sita G.; Romasco J.; Geibel C.; Lammerhofer M.; Goettert M.I.; Tarozzi A.; Laufer S.A.; Koch P., Discovery and evaluation of enantiopure 9H-pyrimido[4,5‐b]indoles as nanomolar GSK‐3β inhibitors with improved metabolic stability, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2020, 21, Article number: 7823 , pp. 1 - 41 [Scientific article]Open Access

Pruccoli, L; Morroni, F; Sita, G; Hrelia, P; Tarozzi, A, Esculetin as a Bifunctional Antioxidant Prevents and Counteracts the Oxidative Stress and Neuronal Death Induced by Amyloid Protein in SH-SY5Y Cells, «ANTIOXIDANTS», 2020, 9, Article number: 551 , pp. 1 - 16 [Scientific article]Open Access

Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; Ana Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti, Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease, «ACS CHEMICAL NEUROSCIENCE», 2020, 11, pp. 2728 - 2740 [Scientific article]Open Access

Maria Rosa Gigliobianco; Barbara Campisi; Dolores Vargas Peregrina; Roberta Censi; Gulzhan Khamitova; Simone Angeloni; Giovanni Caprioli; Marco Zannotti; Stefano Ferraro; Rita Giovannetti; Cristina Angeloni; Giulio Lupidi; Letizia Pruccoli; Andrea Tarozzi; Dario Voinovich; Piera Di Martino, Optimization of the Extraction from Spent Coffee Grounds Using the Desirability Approach, «ANTIOXIDANTS», 2020, 9, Article number: 370 , pp. 1 - 18 [Scientific article]Open Access

Claudio Viegas Jr; Carlos A Manssour Fraga; Maria Emilia Sousa; Andrea Tarozzi, Oxidative Stress: How Has It Been Considered in the Design of New Drug Candidates for Neurodegenerative Diseases?, «FRONTIERS IN PHARMACOLOGY», 2020, 11, Article number: 609274 , pp. 1 - 3 [Scientific article]Open Access

Andrea Tarozzi, Oxidative Stress in Neurodegenerative Diseases: From Preclinical Studies to Clinical Applications, «JOURNAL OF CLINICAL MEDICINE», 2020, 9, Article number: 1223 , pp. 1 - 4 [Scientific article]Open Access

Vittori, Leydi Natalia; Tarozzi, Andrea; Latessa, Pasqualino Maietta, Circulating Cell-Free DNA in Physical Activities, in: Cell-free DNA as Diagnostic Markers Methods and Protocols, Berlino, Springer, 2019, pp. 183 - 197 (METHODS IN MOLECULAR BIOLOGY) [Chapter or essay]

Emanuela Mhillaj, Andrea Tarozzi, Letizia Pruccoli, Vincenzo Cuomo, Luigia Trabace, Cesare Mancuso, Curcumin and Heme Oxygenase: Neuroprotection and Beyond, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2019, 20, Article number: 2419 , pp. 1 - 11 [Scientific article]Open Access

Simona Sestito, Letizia Pruccoli, Massimiliano Runfola, Valentina Citi, Alma Martelli, Giuseppe Saccomanni, Vincenzo Calderone, Andrea Tarozzi, Simona Rapposell, Design and synthesis of H 2 S-donor hybrids: A new treatment for Alzheimer's disease?, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 184, pp. 1 - 11 [Scientific article]

Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolini M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A., Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 178, pp. 243 - 258 [Scientific article]Open Access

Morroni F.; Sita G.; Graziosi A.; Ravegnini G.; Molteni R.; Paladini M.S.; Dias K.S.T.; Dos Santos A.F.; Viegas C.; Camps I.; Pruccoli L.; Tarozzi A.; Hrelia P., PQM130, a novel feruloyl-donepezil hybrid compound, effectively ameliorates the cognitive impairments and pathology in a mouse model of Alzheimer's disease, «FRONTIERS IN PHARMACOLOGY», 2019, 10, pp. 1 - 16 [Scientific article]Open Access

Heider F.; Pantsar T.; Kudolo M.; Ansideri F.; De Simone A.; Pruccoli L.; Schneider T.; Goettert M.I.; Tarozzi A.; Andrisano V.; Laufer S.A.; Koch P., Pyridinylimidazoles as GSK3β Inhibitors: The Impact of Tautomerism on Compound Activity via Water Networks, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 1407 - 1414 [Scientific article]

Morroni Fabiana, Sita Giulia, Djemil Alice, D'Amico Massimo, Pruccoli Letizia, Cantelli-Forti Giorgio, Hrelia Patrizia, Tarozzi Andrea., Comparison of Adaptive Neuroprotective Mechanisms of Sulforaphane and its Interconversion Product Erucin in in Vitro and in Vivo Models of Parkinson's Disease, «JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY», 2018, 66, pp. 856 - 865 [Scientific article]Open Access