Andreev S.; Pantsar T.; El-gokha A.; Ansideri F.; Kudolo M.; Anton D.B.; Sita G.; Romasco J.; Geibel C.; Lammerhofer M.; Goettert M.I.; Tarozzi A.; Laufer S.A.; Koch P., Discovery and evaluation of enantiopure 9H-pyrimido[4,5‐b]indoles as nanomolar GSK‐3β inhibitors with improved metabolic stability, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2020, 21, Article number: 7823, pp. 1 - 41 [articolo]Open Access
Pruccoli, L; Morroni, F; Sita, G; Hrelia, P; Tarozzi, A, Esculetin as a Bifunctional Antioxidant Prevents and Counteracts the Oxidative Stress and Neuronal Death Induced by Amyloid Protein in SH-SY5Y Cells, «ANTIOXIDANTS», 2020, 9, Article number: 551, pp. 1 - 16 [articolo]Open Access
Rita Maria Concetta Di Martino; Letizia Pruccoli; Alessandra Bisi; Silvia Gobbi; Angela Rampa; Ana Martinez; Concepción Pérez; Loreto Martinez-Gonzalez; Maria Paglione; Elia Di Schiavi; Francesca Seghetti; Andrea Tarozzi; Federica Belluti, Novel Curcumin-Diethyl Fumarate Hybrid as a Dualistic GSK-3β Inhibitor/Nrf2 Inducer for the Treatment of Parkinson's Disease, «ACS CHEMICAL NEUROSCIENCE», 2020, 11, pp. 2728 - 2740 [articolo]Open Access
Rosa Gigliobianco, Maria; Campisi, Barbara; Vargas Peregrina, Dolores; Censi, Roberta; Khamitova, Gulzhan; Angeloni, Simone; Caprioli, Giovanni; Zannotti, Marco; Ferraro, Stefano; Giovannetti, Rita; Angeloni, Cristina; Lupidi, Giulio; Pruccoli, Letizia; Tarozzi, Andrea; Voinovich, Dario; Di Martino, Piera, Optimization of the Extraction from Spent Coffee Grounds Using the Desirability Approach, «ANTIOXIDANTS», 2020, 9, Article number: 370, pp. 1 - 18 [articolo]Open Access
Claudio Viegas Jr; Carlos A Manssour Fraga; Maria Emilia Sousa; Andrea Tarozzi, Oxidative Stress: How Has It Been Considered in the Design of New Drug Candidates for Neurodegenerative Diseases?, «FRONTIERS IN PHARMACOLOGY», 2020, 11, Article number: 609274, pp. 1 - 3 [articolo]Open Access
Andrea Tarozzi, Oxidative Stress in Neurodegenerative Diseases: From Preclinical Studies to Clinical Applications, «JOURNAL OF CLINICAL MEDICINE», 2020, 9, Article number: 1223, pp. 1 - 4 [articolo]Open Access
Vittori, Leydi Natalia; Tarozzi, Andrea; Latessa, Pasqualino Maietta, Circulating Cell-Free DNA in Physical Activities, in: Cell-free DNA as Diagnostic Markers Methods and Protocols, Berlino, Springer, 2019, pp. 183 - 197 (METHODS IN MOLECULAR BIOLOGY) [capitolo di libro]
Emanuela Mhillaj, Andrea Tarozzi, Letizia Pruccoli, Vincenzo Cuomo, Luigia Trabace, Cesare Mancuso, Curcumin and Heme Oxygenase: Neuroprotection and Beyond, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2019, 20, Article number: 2419, pp. 1 - 11 [articolo]Open Access
Montanari S.; Mahmoud A.M.; Pruccoli L.; Rabbito A.; Naldi M.; Petralla S.; Moraleda I.; Bartolini M.; Monti B.; Iriepa I.; Belluti F.; Gobbi S.; Di Marzo V.; Bisi A.; Tarozzi A.; Ligresti A.; Rampa A., Discovery of novel benzofuran-based compounds with neuroprotective and immunomodulatory properties for Alzheimer's disease treatment, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 178, pp. 243 - 258 [articolo]Open Access
Morroni F.; Sita G.; Graziosi A.; Ravegnini G.; Molteni R.; Paladini M.S.; Dias K.S.T.; Dos Santos A.F.; Viegas C.; Camps I.; Pruccoli L.; Tarozzi A.; Hrelia P., PQM130, a novel feruloyl-donepezil hybrid compound, effectively ameliorates the cognitive impairments and pathology in a mouse model of Alzheimer's disease, «FRONTIERS IN PHARMACOLOGY», 2019, 10, pp. 1 - 16 [articolo]Open Access
Heider F.; Pantsar T.; Kudolo M.; Ansideri F.; De Simone A.; Pruccoli L.; Schneider T.; Goettert M.I.; Tarozzi A.; Andrisano V.; Laufer S.A.; Koch P., Pyridinylimidazoles as GSK3β Inhibitors: The Impact of Tautomerism on Compound Activity via Water Networks, «ACS MEDICINAL CHEMISTRY LETTERS», 2019, 10, pp. 1407 - 1414 [articolo]
Morroni Fabiana, Sita Giulia, Djemil Alice, D'Amico Massimo, Pruccoli Letizia, Cantelli-Forti Giorgio, Hrelia Patrizia, Tarozzi Andrea., Comparison of Adaptive Neuroprotective Mechanisms of Sulforaphane and its Interconversion Product Erucin in in Vitro and in Vivo Models of Parkinson's Disease, «JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY», 2018, 66, pp. 856 - 865 [articolo]Open Access
Dias Viegas, Flávia Pereira; de Freitas Silva, Matheus; Divino da Rocha, Miguel; Castelli, Maísa Rosa; Riquiel, Mariana Máximo; Machado, Rafael Pereira; Vaz, Sarah Macedo; Simões de Lima, Laís Medeiros; Mancini, Karla Cristine; Marques de Oliveira, Patrícia Cruz; Morais, Élida Parreira; Gontijo, Vanessa Silva; da Silva, Fernanda Motta R.; D'Alincourt da Fonseca Peçanha, Dora; Castro, Newton Gonçalves; Neves, Gilda A.; Giusti-Paiva, Alexandre; Vilela, Fabiana Cardoso; Orlandi, Lidiane; Camps, Ihosvany; Veloso, Márcia Paranho; Leomil Coelho, Luis Felipe; Ionta, Marisa; Ferreira-Silva, Guilherme Álvaro; Pereira, Rodrigo Machado; Dardenne, Laurent E.; Guedes, Isabella Alvim; de Oliveira Carneiro Junior, Wellerson; Quaglio Bellozi, Paula Maria; Pinheiro de Oliveira, Antônio Carlos; Ferreira, Fábio Furlan; Pruccoli, Letizia; Tarozzi, Andrea; Viegas, Claudio*, Design, synthesis and pharmacological evaluation of N-benzyl-piperidinyl-aryl-acylhydrazone derivatives as donepezil hybrids: Discovery of novel multi-target anti-alzheimer prototype drug candidates, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2018, 147, pp. 48 - 65 [articolo]Open Access
Rampa, Angela*; Bartolini, Manuela; Pruccoli, Letizia; Naldi, Marina; Iriepa, Isabel; Moraleda, Ignacio; Belluti, Federica; Gobbi, Silvia; Tarozzi, Andrea; Bisi, Alessandra, Exploiting the chalcone scaffold to develop multifunctional agents for Alzheimer’s disease, «MOLECULES», 2018, 23, Article number: 1902, pp. 1 - 22 [articolo]Open Access
Morroni, Fabiana*; Sita, Giulia; Graziosi, Agnese; Turrini, Eleonora; Fimognari, Carmela; Tarozzi, Andrea; Hrelia, Patrizia, Neuroprotective effect of caffeic acid phenethyl ester in a mouse model of alzheimer's disease involves Nrf2/HO-1 pathway, «AGING AND DISEASE», 2018, 9, pp. 605 - 622 [articolo]Open Access