Foto del docente

Andrea Cavalli

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Coordinator of PhD Programme in Data Science and Computation

Publications

L.Piazzi; A. Cavalli; F. Colizzi; F. Belluti; M. Bartolini; F. Mancini; M. Recanatini; V. Andrisano; A. Rampa, Multi-target-directed coumarin derivatives: hAChE and BAC1 inhibitors as potential anti-Alzheimer compounds, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2008, 18, pp. 423 - 426 [Scientific article]

A. Cavalli; M. L. Bolognesi; A. Minarini; M.Rosini; V. Tumiatti; M. Recanatini; C. Melchiorre, Multi-target-Directed Ligands To Combat Neurodegenerative Diseases, «JOURNAL OF MEDICINAL CHEMISTRY», 2008, 51, pp. 347 - 372 [Scientific article]

Maria Laura Bolognesi; Federica Lizzi; Christian Bergamini; Serena Leone; Romana Fato; Andrea Cavalli, Parallel synthesis and biological evaluation of a small library of 2-phenoxy-1,4-naphthoquinone and 2-phenoxy-1,4-anthraquinone derivatives bearing antitrypanosomal and antileishmanial activity, in: XII Meeting Strutture Eterocicliche nella Ricerca Farmaceutica, Atti, S. L., s. n., 2008, pp. 205 - 205 (atti di: XII Meeting Strutture Eterocicliche nella Ricerca Farmaceutica,, Palermo, 18-21 maggio 2008) [Abstract]

Cavalli A.; Pacetti A.; Recanatini M.; Prandi C.; Scarpi D.; Occhiato E.G., Predicting reactivity and stereoselectivity in the Nazarov reaction: A combined computational and experimental study, «CHEMISTRY-A EUROPEAN JOURNAL», 2008, 14, pp. 9292 - 9304 [Scientific article]

Recanatini M.; Cavalli A., QSAR and pharmacophores for drugs involved in hERG blockage, in: Antitargets. Prediction and prevention of drug side effects, WEINHEIM, Wiley-VCH, 2008, pp. 109 - 126 (Methods and Principles in Medicinal Chemistry) [Chapter or essay]

S. Rizzo; A. Cavalli; L. Ceccarini; F. Belluti; A. Bisi; M. Bartolini; V. Andrisano; M. Recanatini; A. Rampa, SAR and binding mode at the h-AChE active site of pseudo-irreversible inhibitors related to Xanthostigmine, in: XIX National Meeting on Medicinal Chemistry, s.l, s.n, 2008, pp. 219 - 219 (atti di: XIX National Meeting on Medicinal Chemistry, Verona, 14-18 september 2008) [Abstract]

V. Tumiatti; A. Milelli; A. Minarini; M. Rosini; M. L. Bolognesi; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; C. Melchiorre, Structure-Activity Relationships of Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone. 4. Futher Investigation on the Inner Spacer., «JOURNAL OF MEDICINAL CHEMISTRY», 2008, 51, pp. 7308 - 7312 [Scientific article]

V. Tumiatti; A. Milelli; A. Minarini; M. L. Bolognesi; M. Rosini; M. Micco; V. Andrisano; M. Bartolini; F. Mancini; M. Recanatini; A. Cavalli; F. Colizzi; C. Melchiorre, Structure-Activity Relationships of New Acetylcholinesterase Noncovalent Inhibitors Based on a Polyamine Backbone, in: Atti del XIII Meeting Strutture eterocicliche nella ricerca farmaceutica, s.l, s.n, 2008, pp. 207 - 207 (atti di: XIII Meeting Strutture eterocicliche nella ricerca farmaceutica, Palermo, 18-21 Maggio 2008) [Abstract]

A. Cavalli; M. L. Bolognesi, Structure-based design and synthesis of inhibitors of the trypanothione reductase enzyme from Trypanosoma cruzi., in: XIX National Meeting on Medicinal Chemistry, Book of Abstracts, S. L., s. n., 2008, pp. 180 - 180 (atti di: XIX National Meeting on Medicinal Chemistry, Verona, 14-18 Settembre 2008) [Abstract]

Jagusch C.; Negri M.; Hille U.E.; Hu Q.; Bartels M.; Jahn-Hoffmann K.; Pinto-Bazurco Mendieta M.A.; Rodenwaldt B.; Müller-Vieira U.; Schmidt D.; Lauterbach T.; Recanatini M.; Cavalli A.; Hartmann R.W., Synthesis, biological evaluation and molecular modelling studies of methyleneimidazole substituted biaryls as inhibitors of human 17alpha-hydroxylase-17,20-lyase (CYP17). Part I: Heterocyclic modifications of the core structure, «BIOORGANIC & MEDICINAL CHEMISTRY», 2008, 16, pp. 1992 - 2010 [Scientific article]

Bolognesi ML; Lizzi F; Perozzo R; Brun R; Cavalli A., Synthesis of a small library of 2-phenoxy-1,4-naphthoquinone and 2-phenoxy-1,4-anthraquinone derivatives bearing anti-trypanosomal and anti-leishmanial activity, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2008, 18, pp. 2272 - 2276 [Scientific article]

ML. Bolognesi; A. Minarini; M. Bartolini; A. Cavalli; F. Mancini; V. Andrisano; M. Rosini; V. Tumiatti; C. Melchiorre, Synthesis of monomeric derivatives to probe Memoquin bivalent interactions, in: Book of Abstracts, s.l, s.n, 2008, pp. 226 - 226 (atti di: XIX National Meeting on Medicinal Chemistry, Verona, 14-18 September 2008) [Abstract]

Petraglio G.; Bartolini M.; Branduardi D.; Andrisano V.; Recanatini M.; Gervasio F. L.; Cavalli A.; Parrinello M., The role of Li(+), Na(+), and K(+) in the ligand binding inside the human acetylcholinesterase gorge, «PROTEINS», 2008, 70, pp. 779 - 785 [Scientific article]

A. Cavalli; Ml.L. Bolognesi, Two medicinal chemistry approaches to the search for new antitrypanosomal and antileishmanial agents, in: Book of proceedings of the International Conference on Drug Design and Discovery for Developing Countries, TRIESTE, ICS-UNIDO, 2008, pp. XX - YY (atti di: International Conference on Drug Design and Discovery for Developing Countries, Trieste, 3-5 July 2008) [Contribution to conference proceedings]

Cavalli A.; Bolognesi M. L.; Capsoni S.; Andrisano V.; Bartolini M.; Margotti E.; Cattaneo A.; Recanatini M.; Melchiorre C., A small molecule targeting the multifactorial nature of Alzheimer's disease, «ANGEWANDTE CHEMIE. INTERNATIONAL EDITION», 2007, 46, pp. 3689 - 3692 [Scientific article]

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