Foto del docente

Alessandra Locatelli

Professoressa associata

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHEM-07/A Chimica farmaceutica

Delegata del Dipartimento di Farmacia e Biotecnologie

Pubblicazioni

Morigi, R., Locatelli, A., Leoni, A., Rambaldi, M., Bortolozzi, R., Mattiuzzo, E., Ronca, R., Maccarinelli, F., Hamel, E., Bai, R., Brancale, A., Viola, G., Synthesis, in vitro and in vivo biological evaluation of substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones as new potent anticancer agents, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 166, pp. 514 - 530 [articolo]Open Access

Morigi, Rita; Vitali, Beatrice; Prata, Cecilia; Palomino, Rogers A. A; Graziadio, Alessandra; Locatelli, Alessandra; Rambaldi, Mirella; Leoni, Alberto, Investigation on the effects of antimicrobial imidazo[2,1-b]thiazole derivatives on the genitourinary microflora, «MEDICINAL CHEMISTRY», 2018, 14, pp. 311 - 319 [articolo]

R. Morigi, J. Amato, N. Iaccarino, B. Pagano, A. Locatelli, A. Leoni, M. Rambaldi, G. Miglietta, J. Marinello, G. Capranico, E. Novellino, A. Randazzo, Targeting human telomeric and promoter G-quardruplexes: synthesis, biophysical and biological studies of new guanylhydrazones as potential antitumor agents, in: BIONIC 2018: Biology of non-canonical nucleic acids: from humans to pathogens. 26th - 28th September 2018 - Padova, Italy - Abstract Book, Padova, 2018, pp. 126 - 126 (atti di: BIONIC 2018: Biology of non-canonical nucleic acids: from humans to pathogens., Padova, 26-28 settembre 2018) [atti di convegno-abstract]

Leoni, Alberto; Locatelli, Alessandra; Morigi, Rita; Rambaldi, Mirella, A Patent Review on Thiazole Derivatives (2008-2013), «ACTA CHIMICA & PHARMACEUTICA INDICA», 2017, 7, Article number: 103, pp. 1 - 35 [articolo]

Leoni, Alberto; Locatelli, Alessandra; Morigi, Rita; Rambaldi, Mirella, Imidazo[2,1-b] Thiazole: Introduction, Current and Perspective, «BIOENERGETICS», 2017, 6, Article number: Chemistry Journals-17-99R1, pp. 1 - 3 [articolo]

N. Iaccarino, J. Amato, R. Morigi, A. Pagano, A. De Magis, G. Capranico, A. Locatelli, A. Graziadio, A. Leoni, M. Rambaldi, E. Novellino, S. Neidle, B. Pagano, A. Randazzo., Toward the development of specific G-quadruplex binders: biophysical studies of new hydrazone derivatives., in: 6th International Meeting on Quadruplex Nuceic Acids: G4thering. Prague, May 31st-June 3rd, 2017 - Abstract Book, 2017, pp. 132 - 132 (atti di: 6th International Meeting on Quadruplex Nuceic Acids: G4thering., Praga, 31 maggio-03 giugno 2017) [atti di convegno-abstract]

Leoni, Alberto; Locatelli, Alessandra; Morigi, Rita; Rambaldi, Mirella, 2-Indolinone a versatile scaffold for treatment of cancer: A patent review (2008-2014), «EXPERT OPINION ON THERAPEUTIC PATENTS», 2016, 26, pp. 149 - 173 [articolo]

Morigi, Rita; Rambaldi, Mirella; Locatelli, Alessandra; Leoni, Alberto, Small-Molecules Targeting Kinases Involved in Pulmonary Hypertension: a Patent Review (2010-2015), «CURRENT MEDICINAL CHEMISTRY», 2016, 23, pp. 3510 - 3527 [articolo]

Graziadio, Alessandra; Locatelli, Alessandra; Morigi, Rita; Rambaldi, Mirella, Small-Molecules Targeting Sirtuin 1: A Patent Review (2012-2015), «MEDICINAL CHEMISTRY», 2016, 6, pp. 411 - 421 [articolo]

Amato, Jussara; Morigi, Rita; Pagano, Bruno; Pagano, Alessia; Ohnmacht, Stephan; De Magis Alessio; Tiang, Yee-Peng; Capranico, Giovanni; Locatelli, Alessandra; Graziadio, Alessandra; Leoni, Alberto; Rambaldi, Mirella; Novellino, Ettore; Neidle, Stephen; Randazzo, Antonio, Toward the Development of Specific G‑Quadruplex Binders: Synthesis, Biophysical, and Biological Studies of New Hydrazone Derivatives, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 5706 - 5720 [articolo]Open Access

Cappadone, C; Stefanelli, C.; Malucelli, E.; Zini, M.; Onofrillo, C.; Locatelli, A.; Rambaldi, M.; Sargenti, A.; Merolle, L.; Farruggia, G.; Graziadio, A.; Montanaro, L.; Iotti, S., P53-dependent and p53-independent anticancer activity of a new indole derivative in human osteosarcoma cells, «BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS», 2015, 467, pp. 348 - 353 [articolo]

Morigi Rita; Locatelli Alessandra; Leoni Alberto; Mirella Rambaldi, Recent Patents on Thiazole Derivatives Endowed with Antitumor Activity, «RECENT PATENTS ON ANTI-CANCER DRUG DISCOVERY», 2015, 10, pp. 280 - 297 [articolo]

Jussara Amato; Nunzia Iaccarino; Bruno Pagano; Rita Morigi; Alessandra Locatelli; Alberto Leoni; Mirella Rambaldi; Pasquale Zizza; Annamaria Biroccio; Ettore Novellino; Antonio Randazzo, Bis-indole derivatives with antitumor activity turn out to be specific ligands of human telomeric G-quadruplex., «FRONTIERS IN CHEMISTRY», 2014, 2, Article number: 54, pp. 1 - 8 [articolo]

Alberto Leoni;Alessandra Locatelli;Rita Morigi;Mirella Rambaldi, Novel thiazole derivatives: a patent review (2008 – 2012; Part 1), «EXPERT OPINION ON THERAPEUTIC PATENTS», 2014, 24, pp. 201 - 216 [articolo]

Alberto Leoni; Alessandra Locatelli; Rita Morigi; Mirella Rambaldi, Novel thiazole derivatives: a patent review (2008-2012. Part.2), «EXPERT OPINION ON THERAPEUTIC PATENTS», 2014, 24, pp. 759 - 777 [articolo]