Foto del docente

Giovanni Capranico

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: BIO/11 Molecular Biology

Publications

N. Iaccarino, J. Amato, R. Morigi, A. Pagano, A. De Magis, G. Capranico, A. Locatelli, A. Graziadio, A. Leoni, M. Rambaldi, E. Novellino, S. Neidle, B. Pagano, A. Randazzo., Toward the development of specific G-quadruplex binders: biophysical studies of new hydrazone derivatives., in: 6th International Meeting on Quadruplex Nuceic Acids: G4thering. Prague, May 31st-June 3rd, 2017 - Abstract Book, 2017, pp. 132 - 132 (atti di: 6th International Meeting on Quadruplex Nuceic Acids: G4thering., Praga, 31 maggio-03 giugno 2017) [Abstract]

Capranico, Giovanni; Marinello, Jessica; Chillemi, Giovanni, Type I DNA Topoisomerases, «JOURNAL OF MEDICINAL CHEMISTRY», 2017, 60, pp. 2169 - 2192 [Scientific article]

Capranico, G.; Martegani, E.; Musci, G.; Raugei, G.; Russo, T.; Zambrano, N.; Zappavigna, V., Biologia molecolare, Napoli, Edises srl, 2016, pp. 469 . [Research monograph]

Cristini, Agnese; Park, Joon-Hyung; Capranico, Giovanni; Legube, Gaëlle; Favre, Gilles; Sordet, Olivier, DNA-PK triggers histone ubiquitination and signaling in response to DNA double-strand breaks produced during the repair of transcription-blocking topoisomerase I lesions, «NUCLEIC ACIDS RESEARCH», 2016, 44, pp. 1161 - 1178 [Scientific article]Open Access

Marinello, Jessica; Bertoncini, Stefania; Aloisi, Iris; Cristini, Agnese; Tagliazucchi, Guidantonio Malagoli; Forcato, Mattia; Sordet, Olivier; Capranico, Giovanni, Dynamic effects of topoisomerase i inhibition on R-loops and short transcripts at active promoters, «PLOS ONE», 2016, 11, Article number: e0147053 , pp. 1 - 18 [Scientific article]

Amato, Jussara; Morigi, Rita; Pagano, Bruno; Pagano, Alessia; Ohnmacht, Stephan; De Magis Alessio; Tiang, Yee-Peng; Capranico, Giovanni; Locatelli, Alessandra; Graziadio, Alessandra; Leoni, Alberto; Rambaldi, Mirella; Novellino, Ettore; Neidle, Stephen; Randazzo, Antonio, Toward the Development of Specific G‑Quadruplex Binders: Synthesis, Biophysical, and Biological Studies of New Hydrazone Derivatives, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 5706 - 5720 [Scientific article]Open Access

Simonetti, Giorgia; Padella, Antonella; Guadagnuolo, Viviana; Papayannidis, Cristina; Volpato, Francesca; Ottaviani, Emanuela; Formica, Serena; Astolfi, Annalisa; Iacobucci, Ilaria; Capranico, Giovanni; Remondini, Daniel; Martinelli, Giovanni, Gene expression signature of aneuploidy in acute myeloid leukemia, «CANCER RESEARCH», 2014, 74, pp. 2243 - 2243 [Abstract]

Giuseppe Zagotto;Alessandra Gianoncelli;Claudia Sissi;Cristina Marzano;Valentina Gandin;Riccardo Pasquale;Giovanni Capranico;Giovanni Ribaudo;Manlio Palumbo, Novel Ametantrone-Amsacrine Related Hybrids as Topoisomerase IIβ Poisons and Cytotoxic Agents, «ARCHIV DER PHARMAZIE», 2014, 347, pp. 728 - 737 [Scientific article]

Malgorzata N. Drwal;Jessica Marinello;Stefano G. Manzo;Laurence P. G. Wakelin;Giovanni Capranico;Renate Griffith, Novel DNA Topoisomerase IIα Inhibitors from Combined Ligand- and Structure-Based Virtual Screening, «PLOS ONE», 2014, 9, Article number: e114904 , pp. 1 - 16 [Scientific article]

D. Bertozzi;J. Marinello;S. G. Manzo;F. Fornari;L. Gramantieri;G. Capranico, The Natural Inhibitor of DNA Topoisomerase I, Camptothecin, Modulates HIF-1 alpha Activity by Changing miR Expression Patterns in Human Cancer Cells, «MOLECULAR CANCER THERAPEUTICS», 2014, 13, pp. 239 - 248 [Scientific article]

Ruolo editoriale nella rivista «Anti-Cancer Agents in Medicinal Chemistry»

J. Marinello;G. Chillemi;S. Bueno;S. G. Manzo;G. Capranico, Antisense transcripts enhanced by camptothecin at divergent CpG-island promoters associated with bursts of topoisomerase I-DNA cleavage complex and R-loop formation, «NUCLEIC ACIDS RESEARCH», 2013, 41, pp. 10110 - 10123 [Scientific article]

Ruolo editoriale nella rivista «Current Pharmaceutical Design»

Petronzi C; Festa M; Peduto A; Castellano M; Marinello J; Massa A; Capasso A; Capranico G; La Gatta A; De Rosa M; Caraglia M; Filosa R., Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: design, synthesis, and cytotoxic evaluation., «JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH», 2013, 32, Article number: 24 , pp. 1 - 11 [Scientific article]

Simone Pieretti;Jurgen R. Haanstra;Muriel Mazet;Remo Perozzo;Christian Bergamini;Federica Prati;Romana Fato;Giorgio Lenaz;Giovanni Capranico;Reto Brun;Barbara M. Bakker;Paul A. M. Michels;Leonardo Scapozza;Maria Laura Bolognesi;Andrea Cavalli, Naphthoquinone Derivatives Exert Their Antitrypanosomal Activity via a Multi-Target Mechanism, «PLOS NEGLECTED TROPICAL DISEASES», 2013, 7, pp. e2012 - e2023 [Scientific article]

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