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Walter Cabri

Professore ordinario

Dipartimento di Chimica "Giacomo Ciamician"

Settore scientifico disciplinare: CHIM/06 CHIMICA ORGANICA

Pubblicazioni

Hanessian S; Auzzas L; Larsson A; Zhang JB; Giannini G; Gallo G; Ciacci A; Cabri W, Vorinostat-Like Molecules as Structural, Stereochemical, and Pharmacological Tools, «ACS MEDICINAL CHEMISTRY LETTERS», 2010, 1, pp. 70 - 74 [articolo]

Brevetto n. US8383616, Aryl isoxazole compounds with antitumoral Activities.

P. Galletti; A. Quintavalla; C. Ventrici; G. Giannini; W. Cabri; S. Penco; G. Gallo; S. Vincenti; D. Giacomini, Azetidinones as Zinc-Binding Groups to Design Selective HDAC8 Inhibitors, «CHEMMEDCHEM», 2009, 4, pp. 1991 - 2001 [articolo]

Cabri W, Catalysis: The pharmaceutical perspective, «CATALYSIS TODAY», 2009, 140, pp. 2 - 10 [replica/breve intervento]

Giannini G.; Marzi M.; Pezzi R.; Brunetti T.; Battistuzzi G.; Marzo M.D.; Cabri W.; Vesci L.; Pisano C., Corrigendum to "N-Hydroxy-(4-oxime)-cinnamide: A versatile scaffold for the synthesis of novel histone deacetilase (HDAC) inhibitors" [Bioorg. Med. Chem. Lett. 19 (2009) 2346] (DOI:10.1016/j.bmcl.2009.02.029), «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2009, 19, pp. 3694 - 3694 [articolo]

Brevetto n. US8865597, Crystalline(6R,7R)-7-[1,2,4]triazolo-3-yl)-2-[(Z)-trityloxyimino]-acety-lamino)- 3-[(R)-1’-tert-butoxycarbonyl-2-oxo-[1,3’]bipyrrolidinyl-(3E)ylidenemethyl-8-oxo- 5-thia-1-aza-bicyclo[4.2.0]oct-2-ene-2-carboxylic acid benzhydril ester; its manufacturing and use.

Brevetto n. WO2009109504, Enol carbamate derivatives as modulators of fatty Acid Amide Hydrolase.

Giannini G; Marzi M; Di Marzo M; Battistuzzi G; Pezzi R; Brunetti T; Cabri W; Vesci L; Pisano C, Exploring bis-(indolyl)methane moiety as an alternative and innovative CAP group in the design of histone deacetylase (HDAC) inhibitors, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2009, 19, pp. 2840 - 2843 [articolo]

Giannini G; Marzi M; Pezzi R; Brunetti T; Battistuzzi G; Di Marzo M; Cabri W; Vesci L; Pisano C, N-Hydroxy-(4-oxime)-cinnamide: A versatile scaffold for the synthesis of novel histone deacetilase (HDAC) inhibitors, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2009, 19, pp. 2346 - 2349 [replica/breve intervento]

Brevetto n. WO2009138416, OXIME CARBAMOYL DERIVATIVES AS MODULATORS OF FATTY ACID AMIDES HYDROLASE.

Brevetto n. US8664210, Aminooxime derivatives of 2 and/or 4 substitued androstanes and androstenes as medicaments for cardiovascular disorders.

Brevetto n. US8598384, Crystalline Teglicar.

Giannini G; Marzi M; Cabri W; Marastoni E; Battistuzzi G; Vesci L; Pisano C; Beretta GL; De Cesare M; Zunino F, E-ring-modified 7-oxyiminomethyl camptothecins: Synthesis and preliminary in vitro and in vivo biological evaluation, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2008, 18, pp. 2910 - 2915 [replica/breve intervento]

Cabri W, Industrial Synthesis Design With Low Environmental Impact In The Pharma Industry, in: New Methodologies and Techniques for a Sustainable Organic Chemistry, DEU, Springer-Verlag, 2008, pp. 119 - 129 [capitolo di libro]

Brevetto n. US8269007, New cristalline form of 7-dimethoxymethylcamptothecin.

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