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Elisa Uliassi

Ricercatrice a tempo determinato tipo b) (senior)

Dipartimento di Farmacia e Biotecnologie

Settore scientifico disciplinare: CHIM/08 CHIMICA FARMACEUTICA

Pubblicazioni

Chalupova K.; Korabecny J.; Bartolini M.; Monti B.; Lamba D.; Caliandro R.; Pesaresi A.; Brazzolotto X.; Gastellier A.-J.; Nachon F.; Pejchal J.; Jarosova M.; Hepnarova V.; Jun D.; Hrabinova M.; Dolezal R.; Zdarova Karasova J.; Mzik M.; Kristofikova Z.; Misik J.; Muckova L.; Jost P.; Soukup O.; Benkova M.; Setnicka V.; Habartova L.; Chvojkova M.; Kleteckova L.; Vales K.; Mezeiova E.; Uliassi E.; Valis M.; Nepovimova E.; Bolognesi M.L.; Kuca K., Novel tacrine-tryptophan hybrids: Multi-target directed ligands as potential treatment for Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2019, 168, pp. 491 - 514 [articolo]

Ramsay, Rona R; Popovic-Nikolic, Marija R; Nikolic, Katarina; Uliassi, Elisa; Bolognesi, Maria Laura, A perspective on multi-target drug discovery and design for complex diseases, «CLINICAL AND TRANSLATIONAL MEDICINE», 2018, 7, Article number: 3, pp. 1 - 14 [articolo]Open Access

Uliassi, Elisa; Piazzi, Lorna; Belluti, Federica; Mazzanti, Andrea; Kaiser, Marcel; Brun, Reto; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura*, Development of a Focused Library of Triazole-Linked Privileged-Structure-Based Conjugates Leading to the Discovery of Novel Phenotypic Hits against Protozoan Parasitic Infections, «CHEMMEDCHEM», 2018, 13, pp. 678 - 683 [articolo]

Uliassi, Elisa; Fiorani, Giulia; Krauth-Siegel, R. Luise; Bergamini, Christian; Fato, Romana; Bianchini, Giulia; Carlos Menéndez, J.; Molina, Maria Teresa; López-Montero, Eulogio; Falchi, Federico; Cavalli, Andrea; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura*, Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase (TbGAPDH) and Trypanosoma cruzi trypanothione reductase (TcTR) and display trypanocidal activity, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 141, pp. 138 - 148 [articolo]

Gandini, Annachiara; Prati, Federica; Uliassi, Elisa; Bolognesi, Maria L., Drug Discovery Strategies for the Generation of Multitarget Ligands against Neglected Tropical Diseases, in: Drug Selectivity: An Evolving Concept in Medicinal Chemistry, Weinheim, Wiley‐VCH Verlag GmbH & Co. KGaA, 2017, pp. 135 - 159 (METHODS AND PRINCIPLES IN MEDICINAL CHEMISTRY) [capitolo di libro]

Uliassi, Elisa*; Prati, Federica; Bongarzone, Salvatore; Bolognesi, Maria Laura, Medicinal Chemistry of Hybrids for Neurodegenerative Diseases, in: Uliassi, Elisa*, Design of Hybrid Molecules for Drug Development, oxford, Elsevier Inc., 2017, pp. 259 - 277 [capitolo di libro]

Bruno, Stefano; Uliassi, Elisa; Zaffagnini, Mirko; Prati, Federica; Bergamini, Christian; Amorati, Riccardo; Paredi, Gianluca; Margiotta, Marilena; Conti, Paola; Costi, Maria Paola; Kaiser, Marcel; Cavalli, Andrea; Fato, Romana; Bolognesi, Maria Laura, Molecular basis for covalent inhibition of glyceraldehyde-3-phosphate dehydrogenase by a 2-phenoxy-1,4-naphthoquinone small molecule, «CHEMICAL BIOLOGY & DRUG DESIGN», 2017, 89, pp. 1 - 11 [articolo]

Uliassi, Elisa; Gandini, Annachiara; Perone, Rosaria Carmela; Bolognesi, Maria Laura*, Neuroregeneration versus neurodegeneration: Toward a paradigm shift in Alzheimer's disease drug discovery, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 995 - 1013 [articolo]

Jeřábek, Jakub; Uliassi, Elisa; Guidotti, Laura; Korábečný, Jan; Soukup, Ondřej; Sepsova, Vendula; Hrabinova, Martina; Kuča, Kamil; Bartolini, Manuela; Peña-Altamira, Luis Emiliano; Petralla, Sabrina; Monti, Barbara; Roberti, Marinella; Bolognesi, Maria Laura, Tacrine-resveratrol fused hybrids as multi-target-directed ligands against Alzheimer's disease, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 127, pp. 250 - 262 [articolo]

Bolognesi, Maria Laura; Gandini, Annachiara; Prati, Federica; Uliassi, Elisa, From Companion Diagnostics to Theranostics: A New Avenue for Alzheimer's Disease?, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 7759 - 7770 [articolo]

Junker, Anna; Balasubramanian, Ramachandran; Ciancetta, Antonella; Uliassi, Elisa; Kiselev, Evgeny; Martiriggiano, Chiara; Trujillo, Kevin; Mtchedlidze, Giorgi; Birdwell, Leah; Brown, Kyle A.; Harden, T. Kendall; Jacobson, Kenneth A, Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists, «JOURNAL OF MEDICINAL CHEMISTRY», 2016, 59, pp. 6149 - 6168 [articolo]

Brevetto n. PCT Application No. PCT/US2016/053397, TRIAZOLE DERIVATIVES AS P2Y14 RECEPTOR ANTAGONISTS.

Brevetto n. US10683277B2, Triazole derivatives as P2Y14 receptor antagonists.

Kiselev, Evgeny; Balasubramanian, Ramachandran; Uliassi, Elisa; Brown, Kyle A.; Trujillo, Kevin; Katritch, Vsevolod; Hammes, Eva; Stevens, Raymond C.; Harden, T. Kendall; Jacobson, Kenneth A., Design, synthesis, pharmacological characterization of a fluorescent agonist of the P2Y14 receptor, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2015, 25, pp. 4733 - 4739 [articolo]

Santucci, Matteo; Vignudelli, Tatiana; Ferrari, Stefania; Mor, Marco; Scalvini, Laura; Bolognesi, Maria Laura; Uliassi, Elisa; Costi, Maria Paola, The Hippo Pathway and YAP/TAZ-TEAD Protein-Protein Interaction as Targets for Regenerative Medicine and Cancer Treatment, «JOURNAL OF MEDICINAL CHEMISTRY», 2015, 58, pp. 4857 - 4873 [articolo]

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