Foto del docente

Eleonora Diamanti

Junior assistant professor (fixed-term)

Department of Pharmacy and Biotechnology

Academic discipline: CHEM-07/A Pharmaceutical Chemistry

Publications

Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Jörg; Hirsch, Anna K H, Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors, «CHEMMEDCHEM», 2023, 18, pp. e202300346 - 1 [Scientific article]Open Access

Diamanti, Eleonora; Souza, Paulo C T; Setyawati, Inda; Bousis, Spyridon; Gómez, Leticia M; Swier, Lotteke J Y M; Shams, Atanaz; Tsarenko, Aleksei; Stanek, Weronika K; Jäger, Manuel; Marrink, Siewert J; Slotboom, Dirk J; Hirsch, Anna K H, Identification of inhibitors targeting the energy-coupling factor (ECF) transporters, «COMMUNICATIONS BIOLOGY», 2023, 6, pp. 1 - 8 [Scientific article]Open Access

Bousis, Spyridon; Winkler, Steffen; Haupenthal, Jörg; Fulco, Francesco; Diamanti, Eleonora; Hirsch, Anna K H, An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay, «INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES», 2022, 23, pp. 1 - 9 [Scientific article]Open Access

Diamanti, Eleonora; Méndez, María; Ross, Tatjana; Kuttruff, Christian A; Lefranc, Julien; Klingler, Franca-Maria; von Nussbaum, Franz; Jung, Manfred; Gehringer, Matthias, Frontiers in Medicinal Chemistry 2022 Goes Virtual, «CHEMMEDCHEM», 2022, 17, pp. 1 - 13 [Scientific article]

Kiefer, Alexander F; Bousis, Spyridon; Hamed, Mostafa M; Diamanti, Eleonora; Haupenthal, Jörg; Hirsch, Anna K H, Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters, «JOURNAL OF MEDICINAL CHEMISTRY», 2022, 65, pp. 8869 - 8880 [Scientific article]Open Access

Diamanti, Eleonora; Hamed, Mostafa M; Lacour, Antoine; Bravo, Patricia; Illarionov, Boris; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H, Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class, «CHEMMEDCHEM», 2022, 17, pp. 1 - 4 [Scientific article]Open Access

Ropponen, Henni-Karoliina; Diamanti, Eleonora; Siemens, Alexandra; Illarionov, Boris; Haupenthal, Jörg; Fischer, Markus; Rottmann, Matthias; Witschel, Matthias; Hirsch, Anna K H, Assessment of the rules related to gaining activity against Gram-negative bacteria, «RSC MEDICINAL CHEMISTRY», 2021, 12, pp. 593 - 601 [Scientific article]

Drost, M; Diamanti, E; Fuhrmann, K; Goes, A; Shams, A; Haupenthal, J; Koch, M; Hirsch, AKH; Fuhrmann, G, Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor, «PHARMACEUTICS», 2021, 14, pp. 1 - 19 [Scientific article]Open Access

Ropponen, Henni-Karoliina; Bader, Chantal D; Diamanti, Eleonora; Illarionov, Boris; Rottmann, Matthias; Fischer, Markus; Witschel, Matthias; Müller, Rolf; Hirsch, Anna K H, Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity, «CHEMMEDCHEM», 2021, 16, pp. 2089 - 2093 [Scientific article]Open Access

Spyridon Bousis; Inda Setyawati; Eleonora Diamanti; Dirk J. Slotboom; Anna K. H. Hirsch, Energy-Coupling Factor Transporters as Novel Antimicrobial Targets, «ADVANCED THERAPEUTICS», 2019, 2, pp. 1 - 17 [Scientific article]

James, Charlotte A; Yu, Krystle K Q; Gilleron, Martine; Prandi, Jacques; Yedulla, Vijayendar R; Moleda, Zuzanna Z; Diamanti, Eleonora; Khan, Momin; Aggarwal, Varinder K; Reijneveld, Josephine F; Reinink, Peter; Lenz, Stefanie; Emerson, Ryan O; Scriba, Thomas J; Souter, Michael N T; Godfrey, Dale I; Pellicci, Daniel G; Moody, D Branch; Minnaard, Adriaan J; Seshadri, Chetan; Van Rhijn, Ildiko, CD1b Tetramers Identify T Cells that Recognize Natural and Synthetic Diacylated Sulfoglycolipids from Mycobacterium tuberculosis, «CELL CHEMICAL BIOLOGY», 2018, 25, pp. 1 - 42 [Scientific article]

Gierse, Robin Matthias; Redeem, Eswar; Diamanti, Eleonora; Wrenger, Carsten; Groves, Matthew R; Hirsch, Anna Kh, DXS as a target for structure-based drug design, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 1277 - 1294 [Scientific article]

Castellani, Beatrice; Diamanti, Eleonora; Pizzirani, Daniela; Tardia, Piero; Maccesi, Martina; Realini, Natalia; Magotti, Paola; Garau, Gianpiero; Bakkum, Thomas; Rivara, Silvia; Mor, Marco; Piomelli, Daniele, Synthesis and characterization of the first inhibitor ofN-acylphosphatidylethanolamine phospholipase D (NAPE-PLD), «CHEMICAL COMMUNICATIONS», 2017, 53, pp. 12814 - 12817 [Scientific article]

Giusepponi, Maria Elena; Cifani, Carlo; Micioni Di Bonaventura, Maria Vittoria; Mattioli, Laura; Hudson, Alan; Diamanti, Eleonora; Del Bello, Fabio; Giannella, Mario; Mammoli, Valerio; Paoletti, Corinne Dalila; Piergentili, Alessandro; Pigini, Maria; Quaglia, Wilma, Combined Interactions with I1-, I2-Imidazoline Binding Sites and α2-Adrenoceptors To Manage Opioid Addiction, «ACS MEDICINAL CHEMISTRY LETTERS», 2016, 7, pp. 956 - 961 [Scientific article]

Diamanti, E; Bottegoni, G; Goldoni, L; Realini, N; Pagliuca, C; Bertozzi, F; Piomelli, D; Pizzirani, D, Pyrazole-Based Acid Ceramidase Inhibitors: Design, Synthesis, and Structure-Activity Relationships, «SYNTHESIS», 2016, 48, pp. 2739 - 2756 [Scientific article]

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