Foto del docente

Anna Minarini

Full Professor

Department of Pharmacy and Biotechnology

Academic discipline: CHIM/08 Pharmaceutical Chemistry

Head of Scuola di Specializzazione in Farmacia Ospedaliera (nuovo ordinamento)

Publications

Andrea Milelli, Chiara Marchetti, Eleonora Turrini, Elena Catanzaro, Roberta Mazzone, Daniela Tomaselli, Carmela FImognari, Vincenzo Tumiatti, Anna MInarini, Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2018, 28, pp. 1001 - 1004 [Scientific article]

Maria Luisa Di Paolo, Giorgio Cozza, Andrea Milelli, Francesca Zonta, Stefania Sarno, Elirosa Minniti, Michela Rosini, Anna Minarini, Novel targets for “old” polyamine analogues: monoamine oxidases and benextramine derivatives, in: 5th International Conference on Polyamines: Biochemical, Physiological and Clinical Perspectives, 2018, pp. 115 - 115 (atti di: 5th International Conference on Polyamines: Biochemical, Physiological and Clinical Perspectives, Howard Civil Service International House, National Taiwan Ocean University Taipei (Taiwan), September 2nd - 7th, 2018) [Poster]

Ortega, Jose Antonio; Riccardi, Laura; Minniti, Elirosa; Borgogno, Marco; Arencibia, Jose M; Greco, Maria L; Minarini, Anna; Sissi, Claudia; De Vivo, Marco, Pharmacophore Hybridization To Discover Novel Topoisomerase II Poisons with Promising Antiproliferative Activity, «JOURNAL OF MEDICINAL CHEMISTRY», 2018, 61, pp. 1375 - 1379 [Scientific article]Open Access

Oviatt A.A., Kuriappan J.A., Minniti E., Vann K.R. , Onuorah P. , Minarini A., M. De Vivo, Osheroff N., Polyamine-containing etoposide derivatives as poisons of human type II topoisomerases: Differential effects on topoisomerase IIα and IIβ, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2018, 28, pp. 2961 - 2968 [Scientific article]

Minarini, Anna, Farmaci che agiscono sul sistema renina-angiotensina, in: Principi di Chimica Farmaceutica- Foye's, L'Essenziale, Padova, Piccin Nuova Libraria, 2017, pp. 240 - 250 . Opera originale: Autore: T.L. Lemke, S.W. Zito, V.F. Roche, D.A. Williams - Titolo: Essentials of Foye's Principles of Medicinal Chemistry [Book contributions (translation)]

Simoni, Elena; Bartolini, Manuela; Abu, Izuddin F; Blockley, Alix; Gotti, Cecilia; Bottegoni, Giovanni; Caporaso, Roberta; Bergamini, Christian; Andrisano, Vincenza; Cavalli, Andrea; Mellor, Ian R; Minarini, Anna; Rosini, Michela, Multitarget drug design strategy in Alzheimer's disease: focus on cholinergic transmission and amyloid-beta aggregation, «FUTURE MEDICINAL CHEMISTRY», 2017, 9, pp. 953 - 963 [Scientific article]

Milelli, Andrea; Marchetti, Chiara; Greco, Maria Laura; Moraca, Federica; Costa, Giosuè; Turrini, Eleonora; Catanzaro, Elena; Betari, Nibal; Calcabrini, Cinzia; Sissi, Claudia; Alcaro, Stefano; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna, Naphthalene diimide-polyamine hybrids as antiproliferative agents: Focus on the architecture of the polyamine chains, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 128, pp. 107 - 122 [Scientific article]

Alice, Pasini; Chiara, Marchetti; Claudia, Sissi; Marilisa, Cortesi; Emanuele, Giordano; Anna, Minarini; Andrea, Milelli, Novel Polyamine–Naphthalene Diimide Conjugates Targeting Histone Deacetylases and DNA for Cancer Phenotype Reprogramming, «ACS MEDICINAL CHEMISTRY LETTERS», 2017, 8, pp. 1218 - 1223 [Scientific article]Open Access

Minniti, Elirosa; Byl, Jo Ann W.; Riccardi, Laura; Sissi, Claudia; Rosini, Michela; De Vivo, Marco; Minarini, Anna; Osheroff, Neil, Novel xanthone-polyamine conjugates as catalytic inhibitors of human topoisomerase IIα, «BIOORGANIC & MEDICINAL CHEMISTRY LETTERS», 2017, 27, pp. 4687 - 4693 [Scientific article]

Maestri, Valentina; Tarozzi, Andrea; Simoni, Elena; Cilia, Antonio; Poggesi, Elena; Naldi, Marina; Nicolini, Benedetta; Pruccoli, Letizia; Rosini, Michela; Minarini, Anna, Quinazoline based α1-adrenoreceptor antagonists with potent antiproliferative activity in human prostate cancer cell lines, «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2017, 136, pp. 259 - 269 [Scientific article]

Simoni, Elena; Serafini, Melania M; Caporaso, Roberta; Marchetti, Chiara; Racchi, Marco; Minarini, Anna; Bartolini, Manuela; Lanni, Cristina; Rosini, Michela, Targeting the Nrf2/Amyloid-Beta Liaison in Alzheimer's Disease: A Rational Approach, «ACS CHEMICAL NEUROSCIENCE», 2017, 8, pp. 1618 - 1627 [Scientific article]

Tarozzi, A; Marchetti, C; Nicolini, B; D'Amico, M; Ticchi, N; Pruccoli, L; Tumiatti, V; Simoni, E; Lodola, A; Mor, M; Milelli, A; Minarini, A., Combined inhibition of the EGFR/AKT pathways by a novel conjugate of quinazoline with isothiocyanate., «EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY», 2016, 117, pp. 283 - 291 [Scientific article]

Reggiani, Angelo M.; Simoni, Elena; Caporaso, Roberta; Meunier, Johann; Keller, Emeline; Maurice, Tangui; Minarini, Anna; Rosini, Michela; Cavalli, Andrea, In vivo characterization of ARN14140, a memantine/galantamine-based multi-target compound for Alzheimer's disease, «SCIENTIFIC REPORTS», 2016, 6, Article number: 33172 , pp. 1 - 11 [Scientific article]Open Access

Rosini, M; Simoni, E; Caporaso, R; Minarini, A, Multitarget strategies in Alzheimer's disease: benefits and challenges on the road to therapeutics, «FUTURE MEDICINAL CHEMISTRY», 2016, 8, pp. 697 - 711 [Scientific article]

Simoni, Elena; Serafini, Melania M.; Bartolini, Manuela; Caporaso, Roberta; Pinto, Antonella; Necchi, Daniela; Fiori, Jessica; Vincenza, Andrisano; Minarini, Anna; Lanni, Cristina; Rosini, Michela, Nature-Inspired Multifunctional Ligands: Focusing on Amyloid-Based Molecular Mechanisms of Alzheimer’s Disease, «CHEMMEDCHEM», 2016, 11, pp. 1309 - 1317 [Scientific article]Open Access